卡博替尼是一种有效的多受体酪氨酸激酶抑制剂, 抑制VEGFR2,c-Met,Kit,Axl 和 Flt3 的 IC50 分别为0.035,1.3,4.6,7 和 11.3 nM,是用于治疗甲状腺髓样癌的药物,也是肾细胞癌的第二线治疗药物。它是酪氨酸激酶c-Met和VEGFR2的小分子抑制剂,对AXL和RET也有抑制作用。

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1140909-48-3 N-(4-((6,7-Dimethoxyquinolin-4-yl)oxy)phenyl)-N-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide (S)-2-hydroxysuccinate
BD4349941140909-48-399+%
¥257.00250mg常备现货
190728-25-7 4-((6,7-Dimethoxyquinolin-4-yl)oxy)aniline
BD330677190728-25-797%
¥503.0010g常备现货
35654-56-9 4-Chloro-6,7-dimethoxyquinoline
BD1292835654-56-998%
¥224.0025g常备现货
4101-30-8 1-(2-Amino-4,5-dimethoxyphenyl)ethanone
BD02094101-30-896%
¥120.005g常备现货
598-10-7 Cyclopropane-1,1-dicarboxylic acid
BD2772598-10-797%
¥29.005g常备现货
3697-66-3 1-(Ethoxycarbonyl)cyclopropanecarboxylic acid
BD523343697-66-398%
¥169.005g常备现货
849217-48-7 1-((4-Fluorophenyl)carbamoyl)cyclopropanecarboxylic acid
BD214213849217-48-798%
¥51.005g常备现货
1131-62-0 1-(3,4-Dimethoxyphenyl)ethanone
BD820341131-62-098%
¥27.0010g常备现货
1559-02-0 Diethyl 1,1-cyclopropanedicarboxylate
BD114001559-02-095%
¥28.0010g常备现货
4101-32-0 4',5'-Dimethoxy-2'-nitroacetophenone
BD507634101-32-095%
¥796.005g常备现货
849217-60-3 N-(4-Fluorophenyl)-N'-(4-hydroxyphenyl)cyclopropane-1,1-dicarboxamide
BD247352849217-60-395%
¥893.005g常备现货
13425-93-9 6,7-Dimethoxyquinolin-4-ol
BD1303513425-93-998%
¥585.00100g常备现货
190728-24-6 6,7-Dimethoxy-4-(4-nitrophenoxy)quinoline
BD450116190728-24-697%
¥9359.005g
849217-77-2 1-((4-((6,7-Dimethoxyquinolin-4-yl)oxy)phenyl)carbamoyl)cyclopropane-1-carboxylic acid
BD01245375849217-77-298%
¥8639.001g
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