罗拉吡坦是高效选择性具有口服活性的 neurokinin NK1 受体抑制剂,Ki值为0.66 nM,为治疗化疗所致恶心呕吐(CINV)的药物。

清空选项
630-19-3 Pivalaldehyde
BD155460630-19-396% GC
¥106.0025g常备现货
1214741-21-5 (3R,7aR)-3-(tert-butyl)-1-hydroxy-7a-vinyltetrahydropyrrolo[1,2-c]oxazol-5(3H)-one
BD4477541214741-21-597%
¥892.001g常备现货
53990-33-3 (S)-2-(((Benzyloxy)carbonyl)amino)-2-phenylacetic acid
BD1633753990-33-397%
¥993.001kg常备现货
1067-74-9 Methyl 2-(diethoxyphosphoryl)acetate
BD1394181067-74-997%
¥373.00500g常备现货
1779-49-3 Methyltriphenylphosphonium bromide
BD1400041779-49-398%
¥151.00500g常备现货
1125-88-8 Benzaldehyde dimethyl acetal
BD1153741125-88-897%
¥20.0025g常备现货
582-24-1 2-Hydroxy-1-phenylethanone
BD30431582-24-197%
¥157.0025g常备现货
205654-80-4 (2R,4S)-Benzyl 5-oxo-2,4-diphenyloxazolidine-3-carboxylate
BD766678205654-80-498%
¥2401.0025g常备现货
1214741-20-4 (3R,7AR)-3-(tert-butyl)-7a-vinyldihydropyrrolo[1,2-c]oxazole-1,5(3H,6H)-dione
BD4476901214741-20-497%
¥763.001g
530441-95-3 (R)-1-(1-(Bromomethoxy)ethyl)-3,5-bis(trifluoromethyl)benzene
BD294822530441-95-395+%
¥2114.001g
1178515-20-2 (R)-5-((((S)-1-((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)-2-phenylbut-3-en-2-yl)amino)methyl)-5-vinylpyrrolidin-2-one
BD3331431178515-20-295% mix TBC as stabilizer
¥6055.001g
914462-92-3 (5S,8S)-8-(((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)methyl)-8-phenyl-1,7-diazaspiro[4.5]decan-2-one hydrochloride hydrate
BD316105914462-92-395%
¥3362.00100mg
171284-84-7 (3R,7aS)-3-(tert-Butyl)dihydropyrrolo[1,2-c]oxazole-1,5(3H,6H)-dione
BD258812171284-84-795%
¥7507.005g
1214741-14-6 (S)-1-((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)-2-phenylbut-3-en-2-amine fumarate
BD6891531214741-14-697%
¥122.00250mg
1214741-19-1 (3R,7aR)-3-(tert-Butyl)-1,5-dioxohexahydropyrrolo[1,2-c]oxazole-7a-carbaldehyde
BD7489881214741-19-197%
¥459.001g
552292-08-7 (5S,8S)-8-(((R)-1-(3,5-Bis(trifluoromethyl)phenyl)ethoxy)methyl)-8-phenyl-1,7-diazaspiro[4.5]decan-2-one
BD755781552292-08-798%
¥5046.00100mg
1214741-17-9 BENZYL ((S)-1-((R)-1-(3,5-BIS(TRIFLUOROMETHYL)PHENYL)ETHOXY)-2-PHENYLBUT-3-EN-2-YL)CARBAMATE
BD008721531214741-17-995%
¥6370.001g
1