利伐沙班是一种高效的选择性Factor Xa (FXa) 抑制剂,具有强效抗FXa活性 (IC50 为 0.7 nM,Ki 为 0.4 nM),是一种口服抗凝药物(血液稀释剂)。它通常用于预防血液凝块。它是第一个可用的直接活性因子XA抑制剂,它是口服的。

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