鲁拉西酮是多巴胺 D2 和 5-HT7 的拮抗剂,IC50 值分别为 1.68 和 0.495 nM,也是 5-HT1A 受体的部分激动剂,IC50 值为 6.75 nM,是一种非典型抗精神病药。自2010年以来,它已经被FDA批准用于精神分裂症的治疗,并且从2013年开始用于治疗患有双相I障碍的成年人的抑郁症发作。

清空选项
88-98-2 Cyclohex-4-ene-1,2-dicarboxylic acid
BD12267588-98-295%
¥4578.00100g常备现货
110-17-8 Fumaric acid
BD131629110-17-899+%
¥37.00500g常备现货
87691-87-0 3-(1-Piperazinyl)-1,2-benzisothiazole
BD1317987691-87-095%
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2305-32-0 trans-Cyclohexane-1,2-dicarboxylic acid
BD53932305-32-097%
¥29.0010g常备现货
23031-78-9 Benzo[d]isothiazol-3-amine
BD1952523031-78-995%
¥139.00250mg常备现货
71749-03-6 (3aR,7aR)-Hexahydroisobenzofuran-1,3-dione
BD76328371749-03-698%
¥1085.001g常备现货
1687-30-5 Cyclohexane-1,2-dicarboxylic acid
BD530941687-30-595+%
¥517.00100g
367514-88-3 (3aR,4S,7R,7aS)-2-(((1R,2R)-2-((4-(Benzo[d]isothiazol-3-yl)piperazin-1-yl)methyl)cyclohexyl)methyl)hexahydro-1H-4,7-methanoisoindole-1,3(2H)-dione hydrochloride
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77-79-2 3-Sulfolene
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