艾代拉里斯是一种有效的选择性的 p110δ 抑制剂,IC50 为 2.5 nM,比作用于其他I类 PI3K 酶 (抑制 p110α,p110β 和 p110γ; IC50 分别为 820,565 和 89 nM) 选择性高 40 到 300 倍。 它是一种用于治疗某些血液系统恶性肿瘤的药物。该物质起磷酸肌醇3激酶抑制剂的作用;更具体地说,它阻断P110δ,即磷酸肌醇3激酶的δ同工酶。

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870281-86-0 (S)-2-(1-Aminopropyl)-5-fluoro-3-phenylquinazolin-4(3H)-one
BD290566870281-86-095%
¥95.00250mg常备现货
434-76-4 2-Amino-6-fluorobenzoic acid
BD20829434-76-497%
¥25.005g常备现货
87-42-3 6-Chloro-7H-purine
BD844987-42-398%
¥170.00100g常备现货
34306-42-8 Boc-Abu-OH
BD3330334306-42-897%
¥532.00500g常备现货
385-02-4 2-Fluoro-6-nitrobenzoic acid
BD10309385-02-497%
¥2779.00500g常备现货
767-69-1 6-Bromo-7H-purine
BD108571767-69-198%
¥773.0025g常备现货
870281-83-7 2-Fluoro-6-nitro-N-phenylbenzamide
BD555918870281-83-797%
¥59.001g常备现货
870281-82-6 (S)-2-(1-((9H-Purin-6-yl)amino)propyl)-5-fluoro-3-phenylquinazolin-4(3H)-one
BD224801870281-82-698%
¥242.00250mg常备现货
73-24-5 Purin-6-amine
BD849273-24-598%
¥186.00500g常备现货
87172-81-4 Ethyl (R)-2-hydroxybutanoate
BD0077429987172-81-497%
¥5841.001g常备现货
870281-84-8 (S)-tert-Butyl (1-(2-fluoro-6-nitro-N-phenylbenzamido)-1-oxobutan-2-yl)carbamate
BD629211870281-84-897%
¥3120.0025g
870281-85-9 (S)-tert-Butyl (1-(5-fluoro-4-oxo-3-phenyl-3,4-dihydroquinazolin-2-yl)propyl)carbamate
BD290565870281-85-998%
¥105.001g
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