卡非佐米是一种 proteasome 的不可逆抑制剂,在 ANBL-6 和 RPMI 8226 细胞中,IC50 值 < 5 nM,是一种抗癌药物,作为选择性蛋白酶体抑制剂。在化学上,它是四肽环氧酮,是环氧霉素的类似物。

清空选项
868540-17-4 (S)-4-methyl-N-((S)-1-(((S)-4-methyl-1-((R)-2-methyloxiran-2-yl)-1-oxopentan-2-yl)amino)-1-oxo-3-phenylpropan-2-yl)-2-((S)-2-(2-morpholinoacetamido)-4-phenylbutanamido)pentanamide
BD292920868540-17-498%
¥1127.00100mg常备现货
100564-78-1 (S)-2-((tert-Butoxycarbonyl)amino)-4-phenylbutanoic acid
BD16102100564-78-197%
¥36.0010g常备现货
3235-69-6 Morpholin-4-yl-acetic acid
BD1403993235-69-698%
¥120.0010g常备现货
247068-82-2 tert-Butyl ((S)-4-methyl-1-((R)-2-methyloxiran-2-yl)-1-oxopentan-2-yl)carbamate
BD301524247068-82-295%
¥481.001g常备现货
6638-79-5 N,O-Dimethylhydroxylamine hydrochloride
BD19586638-79-598%
¥276.00500g常备现货
247068-81-1 (S)-tert-Butyl (2,6-dimethyl-3-oxohept-1-en-4-yl)carbamate
BD304038247068-81-196%
¥1044.0010g常备现货
247068-85-5 (S)-2-Amino-4-methyl-1-((R)-2-methyloxiran-2-yl)pentan-1-one 2,2,2-trifluoroacetate
BD304039247068-85-595+%
¥1798.005g常备现货
868540-15-2 (6S,9S,12S)-Benzyl 12-benzyl-9-isobutyl-2,2-dimethyl-4,7,10-trioxo-6-phenethyl-3-oxa-5,8,11-triazatridecan-13-oate
BD304041868540-15-295%
¥142.001g常备现货
557-93-7 2-Bromopropene
BD34099557-93-799%
¥29.005g常备现货
87694-50-6 (S)-N-Methyl-N-methoxy-2-(tert-butoxycarbonylamino)-4-methylpentanamide
BD11826287694-50-698%
¥4251.00100g常备现货
2577-90-4 (S)-Methyl 2-amino-3-phenylpropanoate
BD2253752577-90-497%
¥1449.0010g常备现货
13139-15-6 Boc-L-Leucine
BD22563113139-15-698%
¥32.0025g
5874-73-7 (S)-Methyl 2-((S)-2-((tert-butoxycarbonyl)amino)-4-methylpentanamido)-3-phenylpropanoate
BD2906925874-73-798%
¥2110.001g
90072-18-7 (S)-Methyl 2-((S)-2-amino-4-methylpentanamido)-3-phenylpropanoate 2,2,2-trifluoroacetate
BD44758890072-18-796%
¥1652.001g
868539-96-2 (6S,9S,12S)-Methyl 12-benzyl-9-isobutyl-2,2-dimethyl-4,7,10-trioxo-6-phenethyl-3-oxa-5,8,11-triazatridecan-13-oate
BD627718868539-96-298%
¥9134.0025g
868540-16-3 (S)-2-((S)-4-Methyl-2-((S)-2-(2-morpholinoacetamido)-4-phenylbutanamido)pentanamido)-3-phenylpropanoic acid
BD303674868540-16-398%
¥7859.005g
1140908-89-9 (S)-Methyl 2-((S)-4-methyl-2-((S)-2-(2-morpholinoacetamido)-4-phenylbutanamido)pentanamido)-3-phenylpropanoate
BD7666891140908-89-998%
¥9797.0025g
70637-26-2 benzyl (tert-butoxycarbonyl)-L-leucyl-L-phenylalaninate
BD0078230870637-26-298%
¥6026.001g
962-39-0 (S)-Benzyl 2-amino-3-phenylpropanoate
BD00739921962-39-095%
¥719.00100g
70637-28-4 (S)-benzyl 2-((S)-2-amino-4-methylpentanamido)-3-phenylpropanoate 2,2,2-trifluoroacetate
BD0081349970637-28-498%
¥3506.001g
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