培马贝特是过氧化物酶体增殖物激活受体α(PPARα)激动剂,对 h-PPARα,h-PPARγ 和 h-PPARδ 的 EC50 值分别为 1 nM,1.10 μM 和 1.58 μM,是一种降血脂剂。

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