硼替佐米是有效的 20S 蛋白酶体 (20S proteasome) 抑制剂,Ki 为 0.6 nM,是一种抗肿瘤药物,是人类应用的第一种治疗性蛋白酶体抑制剂。蛋白酶体是分解蛋白质的细胞复合物。在一些癌症中,通常杀死癌细胞的蛋白质被分解得太快。硼替佐米阻断了这一过程,并让这些蛋白质杀死癌细胞。在美国和欧洲被批准用于治疗复发性多发性骨髓瘤和套细胞淋巴瘤。

清空选项
1243174-57-3 (R)-3-Methyl-1-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)butan-1-amine hydrochloride
BD2897331243174-57-395%
¥1012.00250mg常备现货
201733-56-4 5,5,5',5'-Tetramethyl-2,2'-bi(1,3,2-dioxaborinane)
BD12402201733-56-498%
¥15.005g常备现货
84110-40-7 Isobutylboronic acid
BD866684110-40-798%
¥417.00100g常备现货
67562-20-3 2-Isobutyl-4,4,5,5-tetramethyl-1,3,2-dioxaborolane
BD23626967562-20-397%
¥75.005g常备现货
18680-27-8 (1S,2S,3R,5S)-2,6,6-Trimethylbicyclo[3.1.1]heptane-2,3-diol
BD1903818680-27-897%
¥39.005g常备现货
179324-69-7 ((R)-3-Methyl-1-((S)-3-phenyl-2-(pyrazine-2-carboxamido)propanamido)butyl)boronic acid
BD106087179324-69-798%
¥203.00100mg常备现货
98-97-5 Pyrazine-2-carboxylic acid
BD261298-97-598%
¥804.001kg常备现货
73183-34-3 4,4,4',4',5,5,5',5'-Octamethyl-2,2'-bi(1,3,2-dioxaborolane)
BD1430473183-34-398%
¥20.005g常备现货
114457-94-2 (S)-3-Phenyl-2-(pyrazine-2-carboxamido)propanoic acid
BD48966114457-94-298%
¥171.0010g常备现货
7524-50-7 H-Phe-OMe.HCl
BD121747524-50-797%
¥73.00100g常备现货
2577-90-4 (S)-Methyl 2-amino-3-phenylpropanoate
BD2253752577-90-497%
¥1449.0010g常备现货
13734-34-4 Boc-Phe-OH
BD852913734-34-498%
¥299.00500g常备现货
73058-37-4 4-(8,9-Dihydropyrido[2,3-b]-1,6-naphthyridin-7(6H)-yl)-4-oxobutanoic acid
BD18320873058-37-495%
¥1743.00250mg
179538-58-0 3-Methyl-1-(tetramethyl-1,3,2-dioxaborolan-2-yl)butan-1-amine hydrochloride
BD01039664179538-58-095%
¥11172.001g
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