阿西替尼是一种 VEGFR 抑制剂,高浓度时也抑制 PDGFR,作用于 VEGFR1,VEGFR2,VEGFR3 和 PDGFRβ,IC50 分别为 0.1 nM,0.2 nM,0.1-0.3 nM 和 1.6 nM,是一种小分子酪氨酸激酶抑制剂。

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886230-77-9 (E)-6-Iodo-3-(2-(pyridin-2-yl)vinyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole
BD632939886230-77-998%
¥1097.005g常备现货
4892-02-8 Methyl 2-mercaptobenzoate
BD1058044892-02-897%
¥100.0010g常备现货
20054-45-9 2-Mercapto-N-methylbenzamide
BD16864120054-45-998%
¥29.001g常备现货
261953-36-0 6-Iodo-1H-indazole
BD28210261953-36-098%
¥1401.00100g常备现货
70315-70-7 3-Iodo-6-nitro-1H-indazole
BD8749670315-70-797%
¥809.0025g常备现货
319460-85-0 (E)-N-Methyl-2-((3-(2-(pyridin-2-yl)vinyl)-1H-indazol-6-yl)thio)benzamide
BD114869319460-85-098%
¥179.00100mg常备现货
115666-47-2 6-Iodo-1H-indole
BD173568115666-47-297%
¥1335.0010g常备现货
4363-35-3 (Z/E)-Styrylboronic acid
BD2231754363-35-395%
¥1232.005g常备现货
7597-18-4 6-Nitro-1H-indazole
BD225137597-18-495%
¥74.0025g常备现货
1945-84-2 2-Ethynylpyridine
BD747541945-84-298% (stabilized with 0.01%HQ)
¥33.001g常备现货
885518-80-9 6-Iodo-1H-indazole-3-carbaldehyde
BD447614885518-80-998%
¥4228.001g
944835-85-2 2-((1H-Indazol-6-yl)thio)-N-methylbenzamide
BD450031944835-85-297%
¥2864.001g
886230-76-8 (E)-3-(2-(Pyridin-2-yl)vinyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-6-amine
BD636768886230-76-897% mix TBC as stabilizer
¥3169.0025g
885126-34-1 2-((3-Iodo-1H-indazol-6-yl)thio)-N-methylbenzamide
BD235568885126-34-198+%
¥5153.001g
886230-74-6 3-Iodo-6-nitro-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole
BD245057886230-74-695+%
¥2393.001g
886230-75-7 (E)-6-Nitro-3-(2-(pyridin-2-yl)vinyl)-1-(tetrahydro-2H-pyran-2-yl)-1H-indazole
BD245059886230-75-795% mix TBC as stabilizer
¥3699.001g
885126-35-2 N-Methyl-2-[[3-[(1E)-2-(2-pyridinyl)ethenyl]-1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-6-yl]thio]benzamide
BD00796566885126-35-297%
¥968.00100mg
319472-83-8 1H-indazole, 3-iodo-6-nitro-1-[[2-(trimethylsilyl)ethoxy]methyl]-
BD00944630319472-83-895%
¥3255.001g
73870-22-1 Triphenyl(pyridin-2-ylmethyl)phosphonium bromide
BD0095187573870-22-198%
¥9546.0010g
38700-15-1 Triphenyl(pyridin-2-ylmethyl)phosphonium chloride
BD0092171438700-15-198+%
¥3367.001g
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